Compile Data Set for Download or QSAR
Found 250 Enz. Inhib. hit(s) with all data for entry = 8112
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009366(CHEMBL3233842 | US11504364, Compound Ref.-Comp. | ...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009360(CHEMBL3233835 | US9346814, Cmpd No 23 Example 27)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434163(CHEMBL2385273 | US9346814, Cmpd No 12 Example 15)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM233322(US9346814, Cmpd No 27 Example 32)copy SMILEScopy InChI
Affinity DataIC50: 6.90nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434164(CHEMBL2385272 | US9346814, Cmpd No 13 Example 16)copy SMILEScopy InChI
Affinity DataIC50: 7.10nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009331(CHEMBL3233843 | US9346814, Cmpd No 24 Example 28)copy SMILEScopy InChI
Affinity DataIC50: 8.5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434165(CHEMBL2385271 | US9346814, Cmpd No 11 Example 14)copy SMILEScopy InChI
Affinity DataIC50: 9.20nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434170(CHEMBL2385299 | US9346814, Cmpd No 21 Example 25)copy SMILEScopy InChI
Affinity DataIC50: 9.90nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434166(CHEMBL2385270 | US9346814, Cmpd No 6 Example 9)copy SMILEScopy InChI
Affinity DataIC50: 10.3nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)copy SMILEScopy InChI
Affinity DataIC50: 10.3nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434169(CHEMBL2385300 | US9346814, Cmpd No 22 Example 26)copy SMILEScopy InChI
Affinity DataIC50: 11nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434167(CHEMBL2385302 | US9346814, Cmpd No 8 Example 11)copy SMILEScopy InChI
Affinity DataIC50: 12nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434168(CHEMBL2385301 | US9346814, Cmpd No 7 Example 10)copy SMILEScopy InChI
Affinity DataIC50: 14nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009358(CHEMBL3233833 | US9346814, Cmpd No 33 Example 38)copy SMILEScopy InChI
Affinity DataIC50: 28nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM233323(US9346814, Cmpd No 29 Example 34)copy SMILEScopy InChI
Affinity DataIC50: 40nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009361(CHEMBL3233837 | US9346814, Cmpd No 25 Example 30)copy SMILEScopy InChI
Affinity DataIC50: 59nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009334(CHEMBL3233554 | US9346814, Cmpd No 4 Example 6)copy SMILEScopy InChI
Affinity DataIC50: 63nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009332(CHEMBL3233836 | US9346814, Cmpd No 26 Example 31)copy SMILEScopy InChI
Affinity DataIC50: 64nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009362(CHEMBL3233838 | US9346814, Cmpd No 25 Example 29)copy SMILEScopy InChI
Affinity DataIC50: 70nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50382283(CHEMBL2022530 | US9346814, Ref. Cmpd No 1 (Example...)copy SMILEScopy InChI
Affinity DataIC50: 110nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM233327(US9346814, Ref Cmpd No 8)copy SMILEScopy InChI
Affinity DataIC50: 130nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434171(CHEMBL2385298 | US9346814, Cmpd No 38 Example 43)copy SMILEScopy InChI
Affinity DataIC50: 160nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434162(CHEMBL2385274 | US9346814, Cmpd No 9 Example 12)copy SMILEScopy InChI
Affinity DataIC50: 190nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009356(CHEMBL3233574 | US9346814, Cmpd No 28 Example 33)copy SMILEScopy InChI
Affinity DataIC50: 200nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009340(CHEMBL3233559 | US9346814, Cmpd No 15 Example 19)copy SMILEScopy InChI
Affinity DataIC50: 220nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009341(CHEMBL3233560 | US9346814, Cmpd No 16 Example 20)copy SMILEScopy InChI
Affinity DataIC50: 270nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009339(CHEMBL3233558 | US9346814, Cmpd No 14 Example 18)copy SMILEScopy InChI
Affinity DataIC50: 290nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434162(CHEMBL2385274 | US9346814, Cmpd No 9 Example 12)copy SMILEScopy InChI
Affinity DataIC50: 350nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434161(CHEMBL2385275 | US9346814, Cmpd No 10 Example 13)copy SMILEScopy InChI
Affinity DataIC50: 360nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434161(CHEMBL2385275 | US9346814, Cmpd No 10 Example 13)copy SMILEScopy InChI
Affinity DataIC50: 370nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434159(CHEMBL2385277 | US9346814, Ref Cmpd No 7 (example ...)copy SMILEScopy InChI
Affinity DataIC50: 420nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM233322(US9346814, Cmpd No 27 Example 32)copy SMILEScopy InChI
Affinity DataIC50: 500nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434166(CHEMBL2385270 | US9346814, Cmpd No 6 Example 9)copy SMILEScopy InChI
Affinity DataIC50: 610nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM233327(US9346814, Ref Cmpd No 8)copy SMILEScopy InChI
Affinity DataIC50: 610nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434176(CHEMBL2385293 | US9346814, Cmpd No 3 Example 4)copy SMILEScopy InChI
Affinity DataIC50: 640nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434176(CHEMBL2385293 | US9346814, Cmpd No 3 Example 4)copy SMILEScopy InChI
Affinity DataIC50: 670nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM233320(US9346814, Ref. Cmpd No 2)copy SMILEScopy InChI
Affinity DataIC50: 670nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434167(CHEMBL2385302 | US9346814, Cmpd No 8 Example 11)copy SMILEScopy InChI
Affinity DataIC50: 710nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009343(CHEMBL3233562 | US9346814, Cmpd No 20 Example 24)copy SMILEScopy InChI
Affinity DataIC50: 750nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434168(CHEMBL2385301 | US9346814, Cmpd No 7 Example 10)copy SMILEScopy InChI
Affinity DataIC50: 840nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)copy SMILEScopy InChI
Affinity DataIC50: 860nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)copy SMILEScopy InChI
Affinity DataIC50: 860nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434163(CHEMBL2385273 | US9346814, Cmpd No 12 Example 15)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009345(CHEMBL3233564 | US9346814, Cmpd No 17 Example 21)copy SMILEScopy InChI
Affinity DataIC50: 1.37E+3nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434164(CHEMBL2385272 | US9346814, Cmpd No 13 Example 16)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009366(CHEMBL3233842 | US11504364, Compound Ref.-Comp. | ...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009342(CHEMBL3233561 | US9346814, Cmpd No 34 Example 39)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50009361(CHEMBL3233837 | US9346814, Cmpd No 25 Example 30)copy SMILEScopy InChI
Affinity DataIC50: 2.03E+3nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM50434189(CHEMBL2385280 | US9346814, Ref. Cmpd No 6 (Example...)copy SMILEScopy InChI
Affinity DataIC50: 2.17E+3nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Universiteit Antwerp; Fox Chase Cancer Center

US Patent
LigandPNGBDBM233328(US9346814, Ref Cmpd No 9)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent
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