Found 62 Enz. Inhib. hit(s) with all data for entry = 8151 TargetProto-oncogene tyrosine-protein kinase Src [251-533,V323S,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 29nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2 [G2019S](Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 45.5nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2 [G2019S](Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 46.9nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2 [G2019S](Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 57.7nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,V323A,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 63nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,V323A,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 67nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2 [G2019S](Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 90.1nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2 [G2019S](Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 100nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 111nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2 [G2019S](Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 121nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2 [G2019S](Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 121nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,V323S,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 131nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 145nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 150nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 186nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 196nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,V323A,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 207nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 213nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 241nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2 [G2019S](Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 274nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 329nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 334nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 334nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 338nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 353nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 380nMAssay Description:In vitro kinase assays using LRRK WT and LRRK G2019S.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 419nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,V323S,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 424nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 560nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 618nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 817nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 899nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 1.00E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 1.00E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 1.66E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 1.76E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 2.17E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 2.32E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 2.76E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 3.08E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 3.16E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 3.50E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
3D Structure (crystal)TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 4.52E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 5.00E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 5.00E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 5.00E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 5.00E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 5.00E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 5.00E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 5.00E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
