Compile Data Set for Download or QSAR
Found 107 Enz. Inhib. hit(s) with all data for entry = 8933
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430058(US10538528, Compound 2)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430053(US10538528, Compound 40)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430052(US10538528, Compound 39)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430054(US10538528, Compound 41)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430066(US10538528, Compound 38)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430051(US10538528, Compound 37)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430029(US10538528, Compound 5)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430064(US10538528, Compound 12)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430030(US10538528, Compound 11)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430063(US10538528, Compound 10)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430062(US10538528, Compound 9)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430061(US10538528, Compound 8)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430060(US10538528, Compound 7)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430070(US10538528, Compound 28)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430037(US10538528, Compound 19)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Akt1 was prepared and assays of inhibitory activity of the compound according to the present invention against Akt1 kinase activity in vitro were con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430056(US10538528, Compound 43)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430057(US10538528, Compound 44)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430072(US10538528, Compound 36)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430065(US10538528, Compound 35)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430050(US10538528, Compound 34)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430047(US10538528, Compound 32)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430041(US10538528, Compound 23)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430031(US10538528, Compound 13)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430059(US10538528, Compound 6)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430068(US10538528, Compound 4)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430067(US10538528, Compound 3)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430028(US10538528, Compound 1)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRyanodine receptor 1 [4317-4329]()
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430056(US10538528, Compound 43)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Rsk1: Inhibitory activity of the compound according to the present invention on Rsk1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430036(US10538528, Compound 18)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Akt1 was prepared and assays of inhibitory activity of the compound according to the present invention against Akt1 kinase activity in vitro were con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430032(US10538528, Compound 14)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Akt1 was prepared and assays of inhibitory activity of the compound according to the present invention against Akt1 kinase activity in vitro were con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRyanodine receptor 1 [4317-4329]()
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430051(US10538528, Compound 37)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Rsk1: Inhibitory activity of the compound according to the present invention on Rsk1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRyanodine receptor 1 [4317-4329]()
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430057(US10538528, Compound 44)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Rsk1: Inhibitory activity of the compound according to the present invention on Rsk1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430045(US10538528, Compound 30)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430037(US10538528, Compound 19)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430049(US10538528, Compound 33)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430055(US10538528, Compound 42)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430069(US10538528, Compound 26)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430042(US10538528, Compound 24)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430038(US10538528, Compound 20)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Akt1 was prepared and assays of inhibitory activity of the compound according to the present invention against Akt1 kinase activity in vitro were con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430038(US10538528, Compound 20)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRyanodine receptor 1 [4317-4329]()
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430053(US10538528, Compound 40)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Rsk1: Inhibitory activity of the compound according to the present invention on Rsk1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRyanodine receptor 1 [4317-4329]()
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430052(US10538528, Compound 39)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Rsk1: Inhibitory activity of the compound according to the present invention on Rsk1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430035(US10538528, Compound 17)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Akt1 was prepared and assays of inhibitory activity of the compound according to the present invention against Akt1 kinase activity in vitro were con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430046(US10538528, Compound 31)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRyanodine receptor 1 [4317-4329]()
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430047(US10538528, Compound 32)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Rsk1: Inhibitory activity of the compound according to the present invention on Rsk1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430039(US10538528, Compound 21)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430035(US10538528, Compound 17)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430034(US10538528, Compound 16)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430033(US10538528, Compound 15)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:S6K1: Inhibitory activity of the compound according to the present invention on S6K1 kinase activity in vitro was assayed using the QSS Assist FP ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
TargetRibosomal protein S6 kinase alpha-1(Homo sapiens (Human))
Taiho Pahrmaceutical Co., Ltd.

US Patent
LigandPNGBDBM430041(US10538528, Compound 23)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Akt1 was prepared and assays of inhibitory activity of the compound according to the present invention against Akt1 kinase activity in vitro were con...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MK6G95US Patent
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