Found 3 Enz. Inhib. hit(s) with Target = '11-beta-hydroxysteroid dehydrogenase 1' and Ligand = 'BDBM50317216'
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Inhibition of human 11-beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Inhibition of mouse 11-beta-HSD1More data for this Ligand-Target Pair
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Pfizer Global Research& Development
Curated by ChEMBL
Pfizer Global Research& Development
Curated by ChEMBL
Affinity DataIC50: 0.320nMAssay Description:Inhibition of human 11-beta-HSD1 expressed in HEK293 cells co-transfected with GRE-luciferase after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair