Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = '11-beta-hydroxysteroid dehydrogenase type 2' and Ligand = 'BDBM29864'
Target11-beta-hydroxysteroid dehydrogenase type 2(Homo sapiens (Human))
The University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM29864(N-(Pyridin-2-yl) arylsulfonamide, 26)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of 11beta-HSD2 (unknown origin) expressed in HEK293 cells using cortisone as substrate measured after 2 hrs in presence of NAD+ by HTRF as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0X43PubMed