Found 11 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A' and Ligand = 'BDBM50011247'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£ di Napoli Federico II
Curated by ChEMBL
Universit£ di Napoli Federico II
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Binding affinity to 5HT1A receptor in Sprague-Dawley rat brain cortex homogenates after 30 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£ di Napoli Federico II
Curated by ChEMBL
Universit£ di Napoli Federico II
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor of rat hippocampus tissue.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£ di Napoli Federico II
Curated by ChEMBL
Universit£ di Napoli Federico II
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Binding affinity of 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£ di Napoli Federico II
Curated by ChEMBL
Universit£ di Napoli Federico II
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Compound was evaluated for inhibiting the binding of [3H]- 8-OH-DPAT to 5-HT1A-receptor from cerebral cortex membranes of ratMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£ di Napoli Federico II
Curated by ChEMBL
Universit£ di Napoli Federico II
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Binding affinity against rat hippocampal 5-hydroxytryptamine 1A (5-HT1A) receptor determined using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£ di Napoli Federico II
Curated by ChEMBL
Universit£ di Napoli Federico II
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Binding affinity at 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in rat brain.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£ di Napoli Federico II
Curated by ChEMBL
Universit£ di Napoli Federico II
Curated by ChEMBL
Affinity DataKi: 6.10nMAssay Description:Binding affinity at 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in rat brain.More data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Displacement of [3H]-5-carboxamidotryptamine from human 5-HT1A receptor expressed in HEK293T cell membranes incubated for 90 mins by scintillation co...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£ di Napoli Federico II
Curated by ChEMBL
Universit£ di Napoli Federico II
Curated by ChEMBL
Affinity DataKi: 8.40nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£ di Napoli Federico II
Curated by ChEMBL
Universit£ di Napoli Federico II
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:In vitro Inhibitory activity tested at 5-hydroxytryptamine 1A receptor binding site in ratMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£ di Napoli Federico II
Curated by ChEMBL
Universit£ di Napoli Federico II
Curated by ChEMBL
Affinity DataIC50: 6.5nMAssay Description:Concentration of compound required to inhibit cortical 5-hydroxytryptamine 1A receptor binding sites in rat brain was evaluatedMore data for this Ligand-Target Pair