Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A' and Ligand = 'BDBM50359421'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataKi: 1.23nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-HT1A receptor in Sprague-Dawley albinus rat cerebral cortex membranes after 15 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataKi: 36.7nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-HT1A receptor in Sprague-Dawley albinus rat cerebral cortex membranes after 15 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataEC50: 16.3nMAssay Description:Agonist activity at human 5HT1A receptor expressed in human HeLa cells assessed as inhibition of forskolin-stimulated cAMP production pretreated 20 m...More data for this Ligand-Target Pair