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Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Arena Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Agonist activity at 5HT2A receptor expressed in HEK cells assessed as inhibition of serotonin-induced inositol phosphate accumulationMore data for this Ligand-Target Pair
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