Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2B' and Ligand = 'BDBM50161649'
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Arena Pharmaceuticals Inc.

Curated by ChEMBL
LigandPNGBDBM50161649((1R,S)-8-trifluoromethyl-2,3,4,5-tetrahydro-1-meth...)copy SMILEScopy InChI
Affinity DataEC50:  794nMAssay Description:Agonist activity at human 5HT2B receptor expressed in HEK293 cells assessed as intracellular IP3 accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q211BPubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Arena Pharmaceuticals Inc.

Curated by ChEMBL
LigandPNGBDBM50161649((1R,S)-8-trifluoromethyl-2,3,4,5-tetrahydro-1-meth...)copy SMILEScopy InChI
Affinity DataEC50:  380nMAssay Description:Effective concentration towards 5-hydroxytryptamine 2C receptors transfected in HEK-293 cells was determined by measuring [3H]-phosphoinositol releas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6Q0GPubMed