Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2C' and Ligand = 'BDBM50301297'
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50301297(2-benzyl-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]az...)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-mesulergine from recombinant human 5-HT2C receptor transfected in Swiss mouse 3T3 cells after 150 mins by scintillation proximit...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H998P2PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50301297(2-benzyl-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]az...)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-mesulergine from recombinant human 5-HT2C receptor transfected in Swiss mouse 3T3 cells after 150 mins by scintillation proximit...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H998P2PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50301297(2-benzyl-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]az...)copy SMILEScopy InChI
Affinity DataEC50:  30nMAssay Description:Agonist activity at recombinant human 5-HT2C receptor transfected in CHOK1 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H998P2PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50301297(2-benzyl-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]az...)copy SMILEScopy InChI
Affinity DataEC50:  31nMAssay Description:Agonist activity at human recombinant 5HT2C receptor expressed in CHO K1 cells assessed as induction of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29C6XHCPubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50301297(2-benzyl-6,7,8,9-tetrahydro-2H-pyridazino[4,3-d]az...)copy SMILEScopy InChI
Affinity DataEC50:  30nMAssay Description:Agonist activity at recombinant human 5-HT2C receptor transfected in CHOK1 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H998P2PubMed