Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2C' and Ligand = 'BDBM50321879' Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University of North Texas Health Science Center
Curated by ChEMBL
University of North Texas Health Science Center
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University of North Texas Health Science Center
Curated by ChEMBL
University of North Texas Health Science Center
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2C receptor using displacement of [3H]DOBMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
F. Hoffmann-La Roche Inc
Curated by ChEMBL
F. Hoffmann-La Roche Inc
Curated by ChEMBL
Affinity DataEC50: 2.00E+3nMAssay Description:Efficacy (pEC50) was evaluated for 5-HT2C receptor-mediated stimulation of IP3 formation in vitro in choroid plexus of the ratMore data for this Ligand-Target Pair
