Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 3A' and Ligand = 'BDBM50060688'
Target5-hydroxytryptamine receptor 3A(RAT)
European Research Centre for Drug Discovery and Development

Curated by ChEMBL
LigandPNGBDBM50060688(7-Fluoro-4-(4-methyl-piperazin-1-yl)-pyrrolo[1,2-a...)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]LY278584 from 5HT3 receptor in rat cortical homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M908K7PubMed
Target5-hydroxytryptamine receptor 3A(RAT)
European Research Centre for Drug Discovery and Development

Curated by ChEMBL
LigandPNGBDBM50060688(7-Fluoro-4-(4-methyl-piperazin-1-yl)-pyrrolo[1,2-a...)copy SMILEScopy InChI
Affinity DataKi:  0.810nMAssay Description:Displacement of [3H]LY278584 from 5HT3 receptor in rat cortical homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H9963MPubMed
Target5-hydroxytryptamine receptor 3A(GUINEA PIG)
European Research Centre for Drug Discovery and Development

Curated by ChEMBL
LigandPNGBDBM50060688(7-Fluoro-4-(4-methyl-piperazin-1-yl)-pyrrolo[1,2-a...)copy SMILEScopy InChI
Affinity DataEC50:  160nMAssay Description:Agonist activity at 5HT3 receptor in voltage-stimulated guinea pig left atrium assessed as positive inotropic potencyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H9963MPubMed