Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 3A' and Ligand = 'BDBM50081969'
Target5-hydroxytryptamine receptor 3A(RAT)
European Research Centre for Drug Discovery and Development

Curated by ChEMBL
LigandPNGBDBM50081969(9-Methyl-4-(4-methyl-piperazin-1-yl)-pyrrolo[1,2-a...)copy SMILEScopy InChI
Affinity DataKi:  0.790nMAssay Description:Displacement of [3H]LY278584 from 5HT3 receptor in rat cortical homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H9963MPubMed
Target5-hydroxytryptamine receptor 3A(RAT)
European Research Centre for Drug Discovery and Development

Curated by ChEMBL
LigandPNGBDBM50081969(9-Methyl-4-(4-methyl-piperazin-1-yl)-pyrrolo[1,2-a...)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]zacopride from 5HT3 receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M908K7PubMed
Target5-hydroxytryptamine receptor 3A(GUINEA PIG)
European Research Centre for Drug Discovery and Development

Curated by ChEMBL
LigandPNGBDBM50081969(9-Methyl-4-(4-methyl-piperazin-1-yl)-pyrrolo[1,2-a...)copy SMILEScopy InChI
Affinity DataKd:  955nMAssay Description:Antagonist activity at 5HT3 receptor in spontaneously beating guinea pig right atrium assessed as inhibition of serotonin-induced maximum response by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H9963MPubMed