Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 3A' and Ligand = 'BDBM50309888'
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50309888(4-(6-Chloro-5-methyloxazolo[4,5-b]pyridin-2-yl)-1,...)copy SMILEScopy InChI
Affinity DataKi:  244nMAssay Description:Displacement of [3H]LY278584 from mouse 5HT3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN66W3PubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Targacept, Inc

Curated by ChEMBL
LigandPNGBDBM50309888(4-(6-Chloro-5-methyloxazolo[4,5-b]pyridin-2-yl)-1,...)copy SMILEScopy InChI
Affinity DataKi:  244nMAssay Description:Binding affinity to 5HT3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32QPPubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Targacept, Inc

Curated by ChEMBL
LigandPNGBDBM50309888(4-(6-Chloro-5-methyloxazolo[4,5-b]pyridin-2-yl)-1,...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Agonist activity at human 5HT3 receptor expressed in human skin epithelial cells assessed as stimulation of calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN66W3PubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Targacept, Inc

Curated by ChEMBL
LigandPNGBDBM50309888(4-(6-Chloro-5-methyloxazolo[4,5-b]pyridin-2-yl)-1,...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of 5HT3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32QPPubMed