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Affinity DataKi: 0.830nMAssay Description:Displacement of [3H]LSD from human 5-HT6 receptor expressed in hamster BHK cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Antagonist activity at human recombinant 5HT6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Antagonist activity at 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Binding affinity to 5HT6R (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Displacement of [3H]Lu AE60157 from rat brain 5-HT6 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Displacement of [3H]Lu AE60157 from rat brain 5-HT6 receptorMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells after 1 hr by microbeta plate reader analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in HEK293 cell membrane measured after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in COS-7 cells assessed as inhibition of 5HT-induced cAMP accumulation preincubated for 7 mins f...More data for this Ligand-Target Pair
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