Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 6' and Ligand = 'BDBM50304000'
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense de Madrid

Curated by ChEMBL
LigandPNGBDBM50304000(4-(4-Methylpiperazin-1-yl)-2-(1-naphthylmethyl)-1H...)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Antagonist activity at human 5HT6 receptor expressed in COS7 cells assessed as inhibition of seratonin-induced cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z320KQPubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense de Madrid

Curated by ChEMBL
LigandPNGBDBM50304000(4-(4-Methylpiperazin-1-yl)-2-(1-naphthylmethyl)-1H...)copy SMILEScopy InChI
Affinity DataKi:  36.2nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z320KQPubMed