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Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Antagonist activity at human recombinant 5HT6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]-LSD from human 5HT6 receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataKi: 0.724nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HeLa cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataKi: 0.776nMAssay Description:Displacement of [125I]SB-258585 from human recombinant 5HT6 receptor using methiothepin after 45 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Antagonist activity at 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense de Madrid
Curated by ChEMBL
Universidad Complutense de Madrid
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Antagonist activity at 5-HT6 receptor (unknown origin) expressed in NG108-15 cells assessed as reduction in cAMP level after 5 mins by BRET assayMore data for this Ligand-Target Pair
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