Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 7' and Ligand = 'BDBM50015198'
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Universit£ degli Studi di Urbino
Curated by ChEMBL
Universit£ degli Studi di Urbino
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]5-HT from human 5-HT7 receptor expressed in HEK293 cells after 30 mins by microbeta counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Universit£ degli Studi di Urbino
Curated by ChEMBL
Universit£ degli Studi di Urbino
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Antagonist activity at human 5-HT7 receptor expressed in CHO cells assessed as inhibition of 5-HT-stimulated cAMP accumulationMore data for this Ligand-Target Pair