Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'ALK tyrosine kinase receptor/Nucleophosmin' and Ligand = 'BDBM50181672'
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation

Curated by ChEMBL
LigandPNGBDBM50181672(5-benzo[1,3]dioxol-5-yl-2-oxo-1,2-dihydro-pyridine...)copy SMILEScopy InChI
Affinity DataIC50: 7.50E+3nMAssay Description:Antiproliferative activity against human NPM-ALK positive anaplastic large cell lymphoma karpas299 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H994T6PubMed
TargetALK tyrosine kinase receptor/Nucleophosmin(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation

Curated by ChEMBL
LigandPNGBDBM50181672(5-benzo[1,3]dioxol-5-yl-2-oxo-1,2-dihydro-pyridine...)copy SMILEScopy InChI
Affinity DataIC50: 1.74E+4nMAssay Description:Antiproliferative activity against murine BaF3 cell line expressing NPM-ALKMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H994T6PubMed