Compile Data Set for Download or QSAR
Found 6 Enz. Inhib. hit(s) with Target = 'AP2-associated protein kinase 1' and Ligand = 'BDBM311287'
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

US Patent
LigandPNGBDBM311287((S)-1-((2′-chloro-4-(difluoromethyl)-5′...)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F191S4US Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

US Patent
LigandPNGBDBM311287((S)-1-((2′-chloro-4-(difluoromethyl)-5′...)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

US Patent
LigandPNGBDBM311287((S)-1-((2′-chloro-4-(difluoromethyl)-5′...)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CF9T6JUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

US Patent
LigandPNGBDBM311287((S)-1-((2′-chloro-4-(difluoromethyl)-5′...)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5XCXUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

US Patent
LigandPNGBDBM311287((S)-1-((2′-chloro-4-(difluoromethyl)-5′...)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 Cl prepared from 15 μl additions of enzyme and substrates (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Z60S4PUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Company

US Patent
LigandPNGBDBM311287((S)-1-((2′-chloro-4-(difluoromethyl)-5′...)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P55QWSUS Patent