Compile Data Set for Download or QSAR
Found 8 Enz. Inhib. hit(s) with Target = 'AP2-associated protein kinase 1' and Ligand = 'BDBM311380'
TargetAP2-associated protein kinase 1(Mus musculus)TBA
LigandPNGBDBM311380((S)-methyl (5-((2-amino-2,4-dimethylpentyl)oxy)-4-...)copy SMILEScopy InChI
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RSPPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM311380((S)-methyl (5-((2-amino-2,4-dimethylpentyl)oxy)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8RSPPubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM311380((S)-methyl (5-((2-amino-2,4-dimethylpentyl)oxy)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P55QWSUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM311380((S)-methyl (5-((2-amino-2,4-dimethylpentyl)oxy)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 Cl prepared from 15 μl additions of enzyme and substrates (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Z60S4PUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM311380((S)-methyl (5-((2-amino-2,4-dimethylpentyl)oxy)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CF9T6JUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM311380((S)-methyl (5-((2-amino-2,4-dimethylpentyl)oxy)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM311380((S)-methyl (5-((2-amino-2,4-dimethylpentyl)oxy)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F191S4US Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM311380((S)-methyl (5-((2-amino-2,4-dimethylpentyl)oxy)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5XCXUS Patent