Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'AP2-associated protein kinase 1' and Ligand = 'BDBM50511399'
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina at Chapel Hill (UNC-CH)

Curated by ChEMBL
LigandPNGBDBM50511399(CHEMBL4542463)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged AAK1 kinase domain (31 to 396 residues) (unknown origin)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of North Carolina at Chapel Hill (UNC-CH)

Curated by ChEMBL
LigandPNGBDBM50511399(CHEMBL4542463)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of tracer K5 binding to N-terminal nano luciferase-fused AAK1 (unknown origin) expressed in HEK293 cells incubated for 2 hrs followed by N...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed