Affinity DataKi: 250nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 506nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 506+/-111More data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]CPX in guinea pig DDT membrane; 543+/-182More data for this Ligand-Target Pair