Compile Data Set for Download or QSAR
Found 6 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50267577'
TargetAdenosine receptor A1(GUINEA PIG)
Kyowa Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50267577(CHEMBL489640 | N6-((+/-)-endo-norborn-2-yl)adenosi...)copy SMILEScopy InChI
Affinity DataKi:  0.320nMAssay Description:Binding affinity against adenosine A1 receptor using N6-[3H]cyclohexyladenosine as radioligand in guinea pig forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NS0VJZPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50267577(CHEMBL489640 | N6-((+/-)-endo-norborn-2-yl)adenosi...)copy SMILEScopy InChI
Affinity DataKi:  0.420nMAssay Description:Binding affinity against Adenosine A1 receptor using [3H]CHA in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TX3FZFPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50267577(CHEMBL489640 | N6-((+/-)-endo-norborn-2-yl)adenosi...)copy SMILEScopy InChI
Affinity DataKi:  0.540nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C8296ZPubMed
TargetAdenosine receptor A1(GUINEA PIG)
Kyowa Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50267577(CHEMBL489640 | N6-((+/-)-endo-norborn-2-yl)adenosi...)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Inhibition of N6-[3H]cyclohexyladenosine binding to guinea pig forebrain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NS0VJZPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50267577(CHEMBL489640 | N6-((+/-)-endo-norborn-2-yl)adenosi...)copy SMILEScopy InChI
Affinity DataKi:  0.910nMAssay Description:Binding affinity against Adenosine A1 receptor using N6-[3H]cyclohexyladenosine in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NS0VJZPubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50267577(CHEMBL489640 | N6-((+/-)-endo-norborn-2-yl)adenosi...)copy SMILEScopy InChI
Affinity DataKi:  0.910nMAssay Description:Binding affinity against Adenosine A1 receptor using N6-[3H]cyclohexyladenosine in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NS0VJZPubMed