Affinity DataKi: 398nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Negative chronotropic activity for A1 Adenosine receptor in spontaneously beating rat atriaMore data for this Ligand-Target Pair
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