TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataKi: 1.36E+3nMAssay Description:Displacement [3H]-CGS-21,680 from Adenosine A2A receptor in rat striatal membrane.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataKi: 1.36E+3nMAssay Description:Displacement [3H]-CGS-21,680 from Adenosine A2A receptor in rat striatal membrane.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute of Diabetes
Curated by ChEMBL
National Institute of Diabetes
Curated by ChEMBL
Affinity DataKi: 1.36E+3nMAssay Description:Affinity at Adenosine A2A receptor in rat striatal membranes by [3H]- CGS 21680 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 5.43E+4nMAssay Description:Binding affinity for HA-tagged mutant human Adenosine A2A receptor (H250N) using [3H]-CGS-21,680 as radioligand expressed in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.26E+4nMAssay Description:Binding affinity for HA-tagged mutant human Adenosine A2A receptor (V84L), using [3H]CGS-21680 as radioligand expressed in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.06E+5nMAssay Description:Binding affinity for HA-tagged wild type human Adenosine A2A receptor (WT) using [3H]CGS-21680 as radioligand expressed in COS-7 cellsMore data for this Ligand-Target Pair
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