TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Trieste
Curated by ChEMBL
Università degli Studi di Trieste
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Displacement of [3H]-ZM-241,385 from human adenosine A2A receptors expressed in HEK-293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Trieste
Curated by ChEMBL
Università degli Studi di Trieste
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Displacement of specific [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Trieste
Curated by ChEMBL
Università degli Studi di Trieste
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]-SCH- 58261 from human adenosine A2A receptor expressed in CHO cells; range 0.22-0.44More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università degli Studi di Trieste
Curated by ChEMBL
Università degli Studi di Trieste
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]-SCH- 58261 from Adenosine A2A receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Inhibition of [3H]-CGS- 21680 binding to Adenosine A2A receptor in rat striatal homogenates.More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Università degli Studi di Ferrara
Curated by ChEMBL
Università degli Studi di Ferrara
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
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