Affinity DataKi: 0.480nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Displacement of [3H]-MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells; range 0.32-0.74More data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:Binding affinity for human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 479nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Inhibition of cAMP accumulation in CHO cells expressing human adenosine A3 receptor; range 3.5-7.6More data for this Ligand-Target Pair
Affinity DataKd: 0.820nMAssay Description:Binding affinity against human Adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair