Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50348163'
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50348163(CHEMBL1800862)copy SMILEScopy InChI
Affinity DataKi:  1.93nMAssay Description:Displacement of [3H]MRE 3008F20 from human adenosine A3 receptor expressed in CHO cells after 120 mins by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N81G6PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50348163(CHEMBL1800862)copy SMILEScopy InChI
Affinity DataIC50: 14.6nMAssay Description:Antagonist activity human adenosine A3 receptor expressed in CHO cells assessed as blockade of Cl-IB-MECA-mediated inhibition of forskolin-stimulated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N81G6PubMed