Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50397717'
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50397717(CHEMBL2181965)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]I-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7HDKPubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50397717(CHEMBL2181965)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in CHO cells by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7HDKPubMed