Compile Data Set for Download or QSAR
Found 6 Enz. Inhib. hit(s) with Target = 'Alpha-2C adrenergic receptor' and Ligand = 'BDBM50419878'
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataKi:  275nMAssay Description:Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2C expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZKTPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataKi:  275nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataKi:  275nMAssay Description:Displacement of [3H]RX821002 from human alpha2C adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3FK6PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataEC50:  2nMAssay Description:Agonist activity at human alpha2C ARMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H134ZZPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataEC50:  2nMAssay Description:Agonist activity at human alpha2C adrenoreceptor expressed in CHO cells assessed as extracellular acidification measured after 4 mins by cytosensor m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3FK6PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universit£ degli Studi di Camerino

Curated by ChEMBL
LigandPNGBDBM50419878(CHEMBL1956195)copy SMILEScopy InChI
Affinity DataEC50:  2nMAssay Description:Agonist activity at human adrenoceptor aplha 2C expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZKTPubMed