Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-ketoglutarate-dependent dioxygenase FTO' and Ligand = 'BDBM50303763'
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Homo sapiens (Human))TBA
LigandPNGBDBM50303763((R)-2-(1-chloro-4-hydroxyisoquinoline-3-carboxamid...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+5nMMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-ketoglutarate-dependent dioxygenase FTO(Homo sapiens (Human))TBA
LigandPNGBDBM50303763((R)-2-(1-chloro-4-hydroxyisoquinoline-3-carboxamid...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of human hexahistidine-tagged full-length FTO expressed in Escherichia coli BL21 (DE3) using 3-methylthymidine as substrate assessed as in...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GBQPubMed