Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A' and Ligand = 'BDBM50155773'
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Oryzon Genomics S.A.

US Patent
LigandPNGBDBM50155773(CHEMBL3781751 | US9469597, 5)copy SMILEScopy InChI
Affinity DataKi: >4.00E+4nM ΔG°: >-26.1kJ/molepH: 7.5 T: 2°CAssay Description:In order to monitor MAO enzymatic activities and/or their inhibition rate by inhibitor(s) of interest, a fluorescence-based (inhibitor)-screening ass...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZW1JVGUS Patent
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Oryzon Genomics S.A.

US Patent
LigandPNGBDBM50155773(CHEMBL3781751 | US9469597, 5)copy SMILEScopy InChI
Affinity DataIC50: 4.13E+4nMAssay Description:Inhibition of recombinant human MAOA incubated for 15 mins measured after 30 mins by luminescence-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22809VXPubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Oryzon Genomics S.A.

US Patent
LigandPNGBDBM50155773(CHEMBL3781751 | US9469597, 5)copy SMILEScopy InChI
Affinity DataIC50: 4.84E+4nMAssay Description:Inhibition of human recombinant MAOA expressed in Pichia pastoris preincubated for 15 mins measured after 30 mins by bioluminescent-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2086767PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Oryzon Genomics S.A.

US Patent
LigandPNGBDBM50155773(CHEMBL3781751 | US9469597, 5)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMpH: 7.5 T: 2°CAssay Description:In order to monitor MAO enzymatic activities and/or their inhibition rate by inhibitor(s) of interest, a fluorescence-based (inhibitor)-screening ass...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZW1JVGUS Patent