BindingDB PrimarySearch

Found 1 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM18166'

Androgen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Company

BDBM18166((6S)-6-hydroxy-2-(4-nitronaphthalen-1-yl)-hexahydr...)copy SMILEScopy InChI

Ki: 4.30nM ΔG°: -47.3kJ/mole EC50: 265nMpH: 7.4 T: 2°CAssay Description:Receptor Binding Assay (Ki)-Binding determined through direct displacement of ligand with [3H]-DHT in the MDA-453 cell line. Transactivation Assay (E...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

PC cid PC sid Patents Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2862DQ9PubMed