Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM468346'
TargetAndrogen receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM468346(US10806720, Compound 1029 | US11648234, Compound 1...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-MIB from wild-type rat AR LBD measured after 16 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1PHBPubMed
TargetAndrogen receptor(Homo sapiens (Human))
University of Tennessee Research Foundation

US Patent
LigandPNGBDBM468346(US10806720, Compound 1029 | US11648234, Compound 1...)copy SMILEScopy InChI
Affinity DataIC50: 2.12E+3nMAssay Description:Methods: hAR-LBD (633-919) was cloned into pGex4t.1. Large scale GST-tagged AR-LBD was prepared and purified using a GST column. Recombinant AR-LBD w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X89PKUS Patent
TargetAndrogen receptor(Homo sapiens (Human))
University of Tennessee Research Foundation

US Patent
LigandPNGBDBM468346(US10806720, Compound 1029 | US11648234, Compound 1...)copy SMILEScopy InChI
Affinity DataIC50: 2.12E+3nMAssay Description:Antagonist activity at recombinant human AR expressed in HEK293 cells assessed as inhibition of R1881-induced transcriptional activity measured after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1PHBPubMed