Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM50215709'
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50215709(CHEMBL1170 | Propionic acid (8R,9S,10R,13S,14S,17S...)copy SMILEScopy InChI
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]DHT from human androgen receptor in MDA453 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9HZ9PubMedDrugBank
TargetAndrogen receptor(Rattus norvegicus (Rat))
University of Basel

Curated by ChEMBL
LigandPNGBDBM50215709(CHEMBL1170 | Propionic acid (8R,9S,10R,13S,14S,17S...)copy SMILEScopy InChI
Affinity DataIC50: 1.91E+3nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CBZPubMed
TargetAndrogen receptor(Mus musculus)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50215709(CHEMBL1170 | Propionic acid (8R,9S,10R,13S,14S,17S...)copy SMILEScopy InChI
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at androgen receptor in mouse C2C12 cells by receptor transactivation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9HZ9PubMed