Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM50469124'
TargetAndrogen receptor(Homo sapiens (Human))
Vancouver Prostate Centre (VPC)

Curated by ChEMBL
LigandPNGBDBM50469124(CHEMBL113332)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of full length AR transcriptional activity in human LNCAP cells harboring AR2PB-eGFP construct assessed as reduction in R1881-induced secr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183967PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Vancouver Prostate Centre (VPC)

Curated by ChEMBL
LigandPNGBDBM50469124(CHEMBL113332)copy SMILEScopy InChI
Affinity DataIC50: 232nMAssay Description:Inhibition of R1881-induced full length AR transcriptional activity in human LNCAP cells harboring AR2PB-eGFP construct after 72 hrs by fluorescence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183967PubMed
TargetAndrogen receptor(Homo sapiens (Human))
Vancouver Prostate Centre (VPC)

Curated by ChEMBL
LigandPNGBDBM50469124(CHEMBL113332)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of R1881-induced transcriptional activity of human AR V7 truncated mutant expressed in human PC3 cells harboring pGL3-ARR3tk-NLuc after 24...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183967PubMed