Found 4 Enz. Inhib. hit(s) with Target = 'Apelin receptor' and Ligand = 'BDBM50565911' 
Affinity DataKi: 4nMAssay Description:Displacement of [125I] [NIe75, Tyr77]Pyr-apelin-13 from YFP-tagged human APJ receptor expressed in HEK293 cell membranes incubated for 1 hr by gamma ...More data for this Ligand-Target Pair
Affinity DataEC50: 2.80nMAssay Description:Agonist activity at human APJ receptor expressed in HEK293 cells co-expressing Galpha(i1)-RlucII(91) assessed as induction of dissociation of Galpha(...More data for this Ligand-Target Pair
Affinity DataEC50: 94nMAssay Description:Agonist activity at human APJ receptor expressed in HEK293T cells co-expressing PDZ-Rho-Gef-RLucll assessed as induction of Galpha12 effector (PDZ-Rh...More data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonist activity at human APJ receptor expressed in HEK293 cells co-expressing Rlucll-beta-arrestin2 assessed as induction of beta-arrestin2 recruitm...More data for this Ligand-Target Pair
