Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM10007'
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM10007(4-[(6-methoxy-1-benzofuran-2-yl)(1H-1,2,4-triazol-...)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q251437DPubMed
TargetAromatase(Homo sapiens (Human))TBA
LigandPNGBDBM10007(4-[(6-methoxy-1-benzofuran-2-yl)(1H-1,2,4-triazol-...)copy SMILEScopy InChI
Affinity DataIC50: 10nMpH: 7.4 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1,2,6,7-3H ]androstenedione / androstenedione during aromatization. Afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3C76PubMed