Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM50254015'
TargetAromatase(Homo sapiens (Human))
Universidade de Coimbra

Curated by ChEMBL
LigandPNGBDBM50254015(1-(2-(3,4-dichlorophenylthio)-2-(4-methoxyphenyl)e...)copy SMILEScopy InChI
Affinity DataKi:  6.5nMAssay Description:Inhibition of human aromatase-mediated conversion of [1beta3H]androstenedione to estrone by Lineweaver-Burk plot in presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ9080PubMed
TargetAromatase(Homo sapiens (Human))
Universidade de Coimbra

Curated by ChEMBL
LigandPNGBDBM50254015(1-(2-(3,4-dichlorophenylthio)-2-(4-methoxyphenyl)e...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of human aromatase-mediated conversion of [1beta3H]androstenedione to estrone by liquid scintillation counting in presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ9080PubMed