Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM50265443'
TargetAromatase(Homo sapiens (Human))
Universidade de Coimbra

Curated by ChEMBL
LigandPNGBDBM50265443(6-chloro-2-methoxy-N-(pyridin-3-yl)acridin-9-amine...)copy SMILEScopy InChI
Affinity DataKi:  25.5nMAssay Description:Inhibition of human aromatase-mediated conversion of [1beta3H]androstenedione to estrone by Lineweaver-Burk plot in presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ9080PubMed
TargetAromatase(Homo sapiens (Human))
Universidade de Coimbra

Curated by ChEMBL
LigandPNGBDBM50265443(6-chloro-2-methoxy-N-(pyridin-3-yl)acridin-9-amine...)copy SMILEScopy InChI
Affinity DataIC50: 76nMAssay Description:Inhibition of human aromatase-mediated conversion of [1beta3H]androstenedione to estrone by liquid scintillation counting in presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ9080PubMed