Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM8889'
TargetAromatase(Homo sapiens (Human))
UNIVERSITAT DES SAARLANDES

US Patent
LigandPNGBDBM8889(3-(3,4-Dihydronaphthalen-2-yl)pyridine | Dihydrona...)copy SMILEScopy InChI
Affinity DataIC50: 4.07nMpH: 7.4Assay Description:The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445KBNUS Patent
TargetAromatase(Homo sapiens (Human))
UNIVERSITAT DES SAARLANDES

US Patent
LigandPNGBDBM8889(3-(3,4-Dihydronaphthalen-2-yl)pyridine | Dihydrona...)copy SMILEScopy InChI
Affinity DataIC50: 4.07E+3nMAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from 3H-labeled androstenedione during aromatization. After incubation, the re...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2FBSPubMed