Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM9917'
TargetAromatase(Homo sapiens (Human))
Universidade de Coimbra

Curated by ChEMBL
LigandPNGBDBM9917(3-[(S)-(4-bromophenyl)(1H-imidazol-1-yl)methyl]-4H...)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of human aromatase-mediated conversion of [1beta3H]androstenedione to estrone by liquid scintillation counting in presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ9080PubMed
TargetAromatase(Homo sapiens (Human))
Universidade de Coimbra

Curated by ChEMBL
LigandPNGBDBM9917(3-[(S)-(4-bromophenyl)(1H-imidazol-1-yl)methyl]-4H...)copy SMILEScopy InChI
Affinity DataIC50: 290nMpH: 7.4 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta,2beta-3H]testosterone during aromatization. After incubation, the ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9NN9PubMed