Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Aurora kinase A' and Ligand = 'BDBM50193014'
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50193014(CHEMBL3942643 | US11155556, No. 9)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM50193014(CHEMBL3942643 | US11155556, No. 9)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of human Aurora kinase A (E122 to K401 residues) expressed in mammalian expression system by Z'LYTE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P91B0PubMed