Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'B1 bradykinin receptor' and Ligand = 'BDBM50309004'
TargetB1 bradykinin receptor(Homo sapiens (Human))
Jerini AG

Curated by ChEMBL
LigandPNGBDBM50309004((R)-N-(1-(5-(5-chloro-3-fluoro-2-(2-methyl-2H-tetr...)copy SMILEScopy InChI
Affinity DataIC50: 0.140nMAssay Description:Antagonist activity at bradikinin B1 receptor in human IMR90 cells assessed as inhibition of des-Arg-bradykinin-mediated calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8ZH1PubMed