Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Beta-3 adrenergic receptor' and Ligand = 'BDBM25761'
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Universität Würzburg

Curated by PDSP Ki Database
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)copy SMILEScopy InChI
Affinity DataKi:  186nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ57C6PubMedDrugBank
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Universität Würzburg

Curated by PDSP Ki Database
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)copy SMILEScopy InChI
Affinity DataKd:  162nMAssay Description:Antagonist activity at human beta-3 adrenergic receptor expressed in fenoterol-stimulated CHOK1 cells assessed as CRE-SPAP level by fluorescence corr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1SBQPubMedDrugBank
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Universität Würzburg

Curated by PDSP Ki Database
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)copy SMILEScopy InChI
Affinity DataKd:  214nMAssay Description:Displacement of [3H]-CGP 12177 from human beta-3 adrenergic receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1SBQPubMedDrugBank
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Universität Würzburg

Curated by PDSP Ki Database
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)copy SMILEScopy InChI
Affinity DataKd:  117nMAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9TKVPubMedDrugBank