Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Beta-3 adrenergic receptor' and Ligand = 'BDBM86453'
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Universität Würzburg

Curated by PDSP Ki Database
LigandPNGBDBM86453(CAS_73573-87-2 | Formoterol | NSC_3083544)copy SMILEScopy InChI
Affinity DataKi:  8.09E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ57C6PubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Universität Würzburg

Curated by PDSP Ki Database
LigandPNGBDBM86453(CAS_73573-87-2 | Formoterol | NSC_3083544)copy SMILEScopy InChI
Affinity DataEC50:  25nMAssay Description:Agonist activity at human recombinant beta3 receptor assessed as cAMP accumulation by radioimmunoassay and cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32X96PubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Universität Würzburg

Curated by PDSP Ki Database
LigandPNGBDBM86453(CAS_73573-87-2 | Formoterol | NSC_3083544)copy SMILEScopy InChI
Affinity DataEC50:  25nMAssay Description:Agonist activity at human beta3 adrenergic receptor expressed in cells by cAMP accumulation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6DFTPubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Universität Würzburg

Curated by PDSP Ki Database
LigandPNGBDBM86453(CAS_73573-87-2 | Formoterol | NSC_3083544)copy SMILEScopy InChI
Affinity DataEC50:  25nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7R2PPubMed