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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Beta-secretase 1 [1-454]' and Ligand = 'BDBM150699'
Target
Beta-secretase 1 [1-454]
(Homo sapiens (Human))
Vitae Pharmaceutical, Inc.
US Patent
Ligand
BDBM150699
(US8981112, 6 | US9526727, 6 | US9949975, Example 6)
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Affinity Data
IC50: 11nM
pH: 4.4
Assay Description:
The inhibitory activity of compounds was assessed by a fluorescence quench assay of BACE1 activity using commercially available substrate HiLyte Fluo...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
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Ligand Info
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2K936GW
US Patent