Found 1 Enz. Inhib. hit(s) with Target = 'Breakpoint cluster region protein/Tyrosine-protein kinase ABL1' and Ligand = 'BDBM50181670'
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
ChemBridge Research Laboratories and ChemBridge Corporation
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Antiproliferative activity against human BCR-ABL positive chronic myeloid leukemia K562 cell lineMore data for this Ligand-Target Pair