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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Bromodomain testis-specific protein [287-359]' and Ligand = 'BDBM205429'
Target
Bromodomain testis-specific protein [287-359]
(Homo sapiens (Human))
TBA
Ligand
BDBM205429
( (R)-JQ1 (3) | US10407441, Compound (R)-JQ1 | US10...)
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Affinity Data
IC50: 217nM
Assay Description:
Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
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MCE
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2TT4V40
US Patent